59321-0
Ramelteon M-II [Mass/volume] in Urine
Active
Part Description
LP100046-4 Ramelteon M-II
The major metabolite of ramelteon, M-II, is active and has approximately one tenth and one fifth the binding affinity of the parent molecule for the human MT1 and MT2 receptors, respectively, and is 17 - 25-fold less potent than ramelteon in in vitro functional assays. Although the potency of M-II at MT1 and MT2 receptors is lower than the parent drug, M-II circulates at higher concentrations than the parent producing 20 - 100 fold greater mean systemic exposure when compared to ramelteon. M-II has weak affinity for the serotonin 5-HT2B receptor, but no appreciable affinity for other receptors or enzymes. Similar to ramelteon, M-II does not interfere with the activity of a number of endogenous enzymes.
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Source: Wikipedia, Ramelteon M-II
Fully-Specified Name
- Component
- Ramelteon M-II
- Property
- MCnc
- Time
- Pt
- System
- Urine
- Scale
- Qn
- Method
Additional Names
- Short Name
- Ramelteon M-II Ur-mCnc
- Display Name
- Ramelteon M-II (U) [Mass/Vol]
- Consumer Name Alpha Get Info
- Ramelteon M-II, Urine
Basic Attributes
- Class
- DRUG/TOX
- Type
- Laboratory
- First Released
- Version 2.32
- Last Updated
- Version 2.70
- Order vs. Observation
- Both
Language Variants Get Info
Tag | Language | Translation |
---|---|---|
es-ES | Spanish (Spain) | Ramelteon M-II: Synonyms: Cuantitativo |
es-MX | Spanish (Mexico) | Ramelteon M-II: |
et-EE | Estonian (Estonia) | Ramelteoon M2: Synonyms: Juhuslik Kvantitatiivne Uriin |
fr-CA | French (Canada) | Ramelteon M-II: |
fr-FR | French (France) | Rameltéon M-II: |
fr-BE | French (Belgium) | Ramelteon M-II: |
it-IT | Italian (Italy) | Ramelteon M-II: Synonyms: Concentrazione di Massa Livelli farmacologici e tossicologia Punto nel tempo (episodio) |
nl-NL | Dutch (Netherlands) | ramelteon M-II: |
pt-BR | Portuguese (Brazil) | Ramelteon M-II: |
ru-RU | Russian (Russian Federation) | Рамелтеон M-II: Synonyms: Количественный Массовая концентрация Точка во времени; |
tr-TR | Turkish (Turkey) | Ramelteon M-II: |
zh-CN | Chinese (China) | 雷美替胺 M-II: Synonyms: M 型 可用数量表示的; |
Example Units
Unit | Source |
---|---|
ng/mL | Example UCUM Units |
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